Ocrelizumab:RA用藥

Motavizumab:RSV

Zibotentan:Prostate cancer

Atrasentan:前列腺癌、卵巢癌、腦癌

Vismodegib:胰臟癌

Fidexaban、OtamixabanApixabanBetrixabanEdoxabanFondaparinux:凝血因子

Vicriviroc:HIV

Taspoglutide:Type 2 diabetes

Cediranib:終止開發

Semagacestat:Alzheimer’s disease 終止開發

Dimebon:Moderate to severe Alzheimer’s disease 終止開發

pegloticase:商品名Krystexxa,痛風治療用

機轉可以參照這邊:

螢幕快照 2011-04-06 上午2.14.43.png  

新機轉圖會在最近幾週出現

Carfilzomib:多發性骨髓瘤治療

Velaglucerase alfa :高雪氏症

Carglumic acid:急性高血氨

Polidocanol 靜脈硬化劑

Cabazitaxel 前列腺癌

Alcaftadine 過敏性結膜炎

Lurasidone 精神分裂症

Tesamorelin HIV lipodystrophy

Tocilizumab Rheumatoid arthritis

Collagenase clostridium histolyticum (Xiaflex) Dupuytren’s contracture

Alglucosidase alfa Pompe’s disease

IncobotulinumtoxinA (Xeomin) Cervical dystonia and blepharospasm

Hizentra Polyvalent human immunoglobulin G

Alpha1-proteinase inhibitor (Glassia) Emphysema

Sipuleucel-T (Provenge) Prostate cancer

brentuximab 淋巴瘤

Tesamorelin(Egrifta®) 愛滋病患的脂肪代謝不良

Alefacept Plaque psoriasis

Muromonab-cD3 Acute transplant rejection

Golimumab rA, PA and As

Natalizumab Multiple sclerosis

canakinumab cryopyrin-associated periodic syndrome

eculizumab Paroxysmal nocturnal haemoglobinuria

Palivizumab Prevention of rsv infection in children

rilonacept cAPs

Ustekinumab Plaque psoriasis

ruxolitinib JAK tyrosine inhibitor

Lestaurtinib JAK tyrosine inhibitor

Tasocitinib JAK3 tyrosine inhibitor

odanacatib 骨質疏鬆症

amonafide 白血症

necitumumab a next-generation version of cetuximab

iniparib poly (ADP-ribose) polymerase 1 (PARP1) inhibitor

gevokizumab interleukin‐1β (IL‐1β)‐targeted monoclonal antibody

palivizumab respiratory syncytial virus

Eribulin mesylate 晚期乳癌

Panobinostat non-selective HDAC inhibitor

selumetinib MEK inhibitor

Ambrisentan Pulmonary hypertension

Ampakines 阿茲海默症


之後會慢慢再針對這些藥物做介紹或是放進機轉圖內

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